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@ARTICLE{Vergallo:155926,
author = {Vergallo, Andrea and Caraci, Filippo and Cuello, A Claudio
and Lemercier, Pablo and Vellas, Bruno and Giudici, Kelly
Virecoulon and Hampel, Harald and Baldacci, Filippo and
Hänisch, Britta and Haberkamp, Marion and Broich, Karl and
Nisticò, Robert and Emanuele, Enzo and Llavero, Francisco
and Zugaza, José L and Lucía, Alejandro and Giacobini,
Ezio and Lista, Simone},
collaboration = {Initiative, Alzheimer Precision Medicine},
title = {{F}uture avenues for {A}lzheimer's disease detection and
therapy: liquid biopsy, intracellular signaling modulation,
systems pharmacology drug discovery.},
journal = {Neuropharmacology},
volume = {185},
issn = {0028-3908},
address = {Amsterdam [u.a.]},
publisher = {Elsevier Science},
reportid = {DZNE-2021-01080},
pages = {108081},
year = {2021},
abstract = {When Alzheimer's disease (AD) disease-modifying therapies
will be available, global healthcare systems will be
challenged by a large-scale demand for clinical and
biological screening. Validation and qualification of
globally accessible, minimally-invasive, and time-,
cost-saving blood-based biomarkers need to be advanced.
Novel pathophysiological mechanisms (and related candidate
biomarkers) - including neuroinflammation pathways (TREM2
and YKL-40), axonal degeneration (neurofilament light chain
protein), synaptic dysfunction (neurogranin, synaptotagmin,
α-synuclein, and SNAP-25) - may be integrated into an
expanding pathophysiological and biomarker matrix and,
ultimately, integrated into a comprehensive blood-based
liquid biopsy, aligned with the evolving
ATN + classification system and the precision medicine
paradigm. Liquid biopsy-based diagnostic and therapeutic
algorithms are increasingly employed in Oncology
disease-modifying therapies and medical practice, showing an
enormous potential for AD and other brain diseases as well.
For AD and other neurodegenerative diseases, newly
identified aberrant molecular pathways have been identified
as suitable therapeutic targets and are currently
investigated by academia/industry-led $R\&D$ programs,
including the nerve-growth factor pathway in basal forebrain
cholinergic neurons, the sigma1 receptor, and the GTPases of
the Rho family. Evidence for a clinical long-term effect on
cognitive function and brain health span of cholinergic
compounds, drug candidates for repositioning programs, and
non-pharmacological multidomain interventions (nutrition,
cognitive training, and physical activity) is developing as
well. Ultimately, novel pharmacological paradigms, such as
quantitative systems pharmacology-based
integrative/explorative approaches, are gaining momentum to
optimize drug discovery and accomplish effective
pathway-based strategies for precision medicine. This
article is part of the special issue on 'The Quest for
Disease-Modifying Therapies for Neurodegenerative
Disorders'.},
subtyp = {Review Article},
keywords = {Alzheimer Disease: diagnosis / Alzheimer Disease: drug
therapy / Alzheimer Disease: metabolism / Animals /
Anti-Inflammatory Agents: administration $\&$ dosage /
Anti-Inflammatory Agents: metabolism / Drug Discovery:
methods / Drug Discovery: trends / Drug Repositioning:
methods / Drug Repositioning: trends / Forecasting / Humans
/ Intracellular Fluid: drug effects / Intracellular Fluid:
metabolism / Liquid Biopsy: methods / Liquid Biopsy: trends
/ Membrane Glycoproteins: metabolism / Pharmacology,
Clinical: methods / Pharmacology, Clinical: trends /
Receptors, Immunologic: metabolism / Signal Transduction:
drug effects / Signal Transduction: physiology / Systems
Biology: methods / Systems Biology: trends / Alzheimer's
disease (Other) / Blood biomarkers (Other) /
Disease-modifying therapies (Other) / Liquid biopsy (Other)
/ Precision medicine (Other) / Systems pharmacology (Other)},
cin = {AG Hänisch},
ddc = {610},
cid = {I:(DE-2719)1013010},
pnm = {354 - Disease Prevention and Healthy Aging (POF4-354)},
pid = {G:(DE-HGF)POF4-354},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:32407924},
doi = {10.1016/j.neuropharm.2020.108081},
url = {https://pub.dzne.de/record/155926},
}