% IMPORTANT: The following is UTF-8 encoded. This means that in the presence % of non-ASCII characters, it will not work with BibTeX 0.99 or older. % Instead, you should use an up-to-date BibTeX implementation like “bibtex8” or % “biber”. @ARTICLE{Scuteri:156003, author = {Scuteri, Damiana and Cassano, Roberta and Trombino, Sonia and Russo, Rossella and Mizoguchi, Hirokazu and Watanabe, Chizuko and Hamamura, Kengo and Katsuyama, Soh and Komatsu, Takaaki and Morrone, Luigi Antonio and Rombolà, Laura and Adornetto, Annagrazia and Laganà, Annarita S and Corasaniti, Maria Tiziana and Tonin, Paolo and Sakurada, Shinobu and Sakurada, Tsukasa and Nicotera, Pierluigi and Bagetta, Giacinto}, title = {{D}evelopment and {T}ranslation of {N}ano{BEO}, a {N}anotechnology-{B}ased {D}elivery {S}ystem of {B}ergamot {E}ssential {O}il {D}eprived of {F}urocumarins, in the {C}ontrol of {A}gitation in {S}evere {D}ementia.}, journal = {Pharmaceutics}, volume = {13}, number = {3}, issn = {1999-4923}, address = {Basel}, publisher = {MDPI}, reportid = {DZNE-2021-01135}, pages = {379}, year = {2021}, abstract = {Dementia is one of the most common causes of disability worldwide characterized by memory loss, cognitive impairment, and behavioral and psychological symptoms (BPSD), including agitation. Treatment of the latter consists of the off-label use of harmful atypical antipsychotics, though a significant reduction is afforded by pain control. The use of an essential oil endowed with analgesic properties and devoid of toxicity would represent an important option for the management of agitation in dementia. Therefore, the aim of this study was to engineer a nanotechnology delivery system based on solid lipid nanoparticles loaded with bergamot essential oil (BEO) and devised in the pharmaceutical form of an odorless cream (NanoBEO) to confirm its analgesic efficacy for further development and application to control agitation in dementia. BEO has proven strong antinociceptive and anti-allodynic properties and, in its bergapten-free form, it is completely devoid of phototoxicity. NanoBEO has been studied in vivo confirming the previously reported analgesic activity of BEO to which is now added its anti-itching properties. Due to the nanotechnology delivery system, the stability of titrated BEO components is guaranteed. Finally, the latter invention, currently under patent consideration, is smell-devoid allowing efficacy and safety to be established in double-blind clinical trials; until now the latter studies have been impeded in aromatherapy by the strong odor of essential oils. A clinical trial NCT04321889 has been designed to provide information about the efficacy and safety of NanoBEO on agitation and pain in patients suffering from severe dementia.}, keywords = {BPSD (Other) / agitation (Other) / dementia (Other) / essential oil of bergamot (Other) / nanotechnology delivery system (Other) / pain (Other)}, cin = {AG Nicotera}, ddc = {610}, cid = {I:(DE-2719)5000018}, pnm = {351 - Brain Function (POF4-351)}, pid = {G:(DE-HGF)POF4-351}, typ = {PUB:(DE-HGF)16}, pubmed = {pmid:33809385}, pmc = {pmc:PMC7999378}, doi = {10.3390/pharmaceutics13030379}, url = {https://pub.dzne.de/record/156003}, }