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@ARTICLE{Lerche:157806,
author = {Lerche, Stefanie and Schulte, Claudia and Wurster, Isabel
and Machetanz, Gerrit and Roeben, Benjamin and Zimmermann,
Milan and Deuschle, Christian and Hauser, Ann-Kathrin and
Böhringer, Judith and Kragelöh-Mann, Ingeborg and Waniek,
Katharina and Lachmann, Ingolf and Petterson, Xuan-Mai T and
Chiang, Ruby and Park, Hyejung and Wang, Bing and
Liepelt-Scarfone, Inga and Maetzler, Walter and Galasko,
Douglas and Scherzer, Clemens R and Gasser, Thomas and
Mielke, Michelle M and Hutten, Samantha J and Mollenhauer,
Brit and Sardi, S Pablo and Berg, Daniela and Brockmann,
Kathrin},
title = {{T}he {M}utation {M}atters: {CSF} {P}rofiles of {GC}ase,
{S}phingolipids, α-{S}ynuclein in {PDGBA}.},
journal = {Movement disorders},
volume = {36},
number = {5},
issn = {1531-8257},
address = {New York, NY},
publisher = {Wiley},
reportid = {DZNE-2021-01263},
pages = {1216 - 1228},
year = {2021},
abstract = {With pathway-specific trials in PD associated with variants
in the glucocerebrosidase gene (PDGBA ) under way, we need
markers that confirm the impact of genetic variants in
patient-derived biofluids in order to allow patient
stratification merely based on genetics and that might serve
as biochemical read-out for target engagement.To explore
GBA-pathway-specific biomarker profiles cross-sectionally
(TUEPAC-MIGAP, PPMI) and longitudinally (PPMI).We measured
enzyme activity of the lysosomal glucocerebrosidase, CSF
levels of glucosylceramides (upstream substrate of
glucocerebrosidase), CSF levels of ceramides (downstream
product of glucocerebrosidase), lactosylceramides,
sphingosines, sphingomyelin (by-products) and CSF levels of
total α-synuclein in PDGBA patients compared to
$PDGBA_wildtype$ patients.Cross-sectionally in both cohorts
and longitudinally in PPMI: (1) glucocerebrosidase activity
was significantly lower in PDGBA compared to
$PDGBA_wildtype$ . (2) CSF levels of upstream substrates
(glucosylceramides species) were higher in PDGBA compared to
$PDGBA_wildtype$ . (3) CSF levels of total α-synuclein were
lower in PDGBA compared to $PDGBA_wildtype$ . All of these
findings were most pronounced in PDGBA with severe mutations
$(PDGBA_severe$ ). Cross-sectionally in TUEPAC-MIGAP and
longitudinally in PPMI, CSF levels of downstream-products
(ceramides) were higher in $PDGBA_severe$ .
Cross-sectionally in TUEPAC-MIGAP by-products sphinganine
and sphingosine-1-phosphate and longitudinally in PPMI
species of by-products lactosylceramides and sphingomyelin
were higher in $PDGBA_severe$ .These findings confirm that
GBA mutations have a relevant functional impact on biomarker
profiles in patients. Bridging the gap between genetics and
biochemical profiles now allows patient stratification for
clinical trials merely based on mutation status.
Importantly, all findings were most prominent in PDGBA with
severe variants. © 2021 International Parkinson and
Movement Disorder Society.},
keywords = {Glucosylceramidase: genetics / Humans / Mutation: genetics
/ Parkinson Disease: genetics / Sphingolipids /
alpha-Synuclein: genetics / CSF (Other) / GBA (Other) /
GCase (Other) / ceramides (Other) / α-synuclein (Other) /
Sphingolipids (NLM Chemicals) / alpha-Synuclein (NLM
Chemicals) / Glucosylceramidase (NLM Chemicals)},
cin = {AG Gasser / AG Berg ; AG Berg / Biobanking Facility
Tübingen / Core ICRU / AG Fischer},
ddc = {610},
cid = {I:(DE-2719)1210000 / I:(DE-2719)5000055 /
I:(DE-2719)1240004 / I:(DE-2719)1240005 /
I:(DE-2719)1410002},
pnm = {353 - Clinical and Health Care Research (POF4-353) / 352 -
Disease Mechanisms (POF4-352)},
pid = {G:(DE-HGF)POF4-353 / G:(DE-HGF)POF4-352},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:33547828},
doi = {10.1002/mds.28472},
url = {https://pub.dzne.de/record/157806},
}