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@ARTICLE{Antn:268494,
author = {Antón, Rosa and Treviño, Miguel Á and Pantoja-Uceda,
David and Félix, Sara and Babu, Maria and Cabrita, Eurico J
and Zweckstetter, Markus and Tinnefeld, Philip and Vera,
Andrés M and Oroz, Javier},
title = {{A}lternative low-populated conformations prompt phase
transitions in polyalanine repeat expansions.},
journal = {Nature Communications},
volume = {15},
number = {1},
issn = {2041-1723},
address = {[London]},
publisher = {Nature Publishing Group UK},
reportid = {DZNE-2024-00240},
pages = {1925},
year = {2024},
abstract = {Abnormal trinucleotide repeat expansions alter protein
conformation causing malfunction and contribute to a
significant number of incurable human diseases. Scarce
structural insights available on disease-related homorepeat
expansions hinder the design of effective therapeutics.
Here, we present the dynamic structure of human PHOX2B
C-terminal fragment, which contains the longest polyalanine
segment known in mammals. The major α-helical conformation
of the polyalanine tract is solely extended by polyalanine
expansions in PHOX2B, which are responsible for most
congenital central hypoventilation syndrome cases. However,
polyalanine expansions in PHOX2B additionally promote
nascent homorepeat conformations that trigger
length-dependent phase transitions into solid condensates
that capture wild-type PHOX2B. Remarkably, HSP70 and HSP90
chaperones specifically seize PHOX2B alternative
conformations preventing phase transitions. The precise
observation of emerging polymorphs in expanded PHOX2B
postulates unbalanced phase transitions as distinct
pathophysiological mechanisms in homorepeat expansion
diseases, paving the way towards the search of therapeutics
modulating biomolecular condensates in central
hypoventilation syndrome.},
keywords = {Animals / Humans / Homeodomain Proteins: metabolism /
Transcription Factors: metabolism / Peptides: genetics /
Peptides: chemistry / Hypoventilation: genetics /
Hypoventilation: congenital / Mutation / Mammals: metabolism
/ Homeodomain Proteins (NLM Chemicals) / polyalanine (NLM
Chemicals) / Transcription Factors (NLM Chemicals) /
Peptides (NLM Chemicals)},
cin = {AG Zweckstetter},
ddc = {500},
cid = {I:(DE-2719)1410001},
pnm = {352 - Disease Mechanisms (POF4-352)},
pid = {G:(DE-HGF)POF4-352},
typ = {PUB:(DE-HGF)16},
pmc = {pmc:PMC10908835},
pubmed = {pmid:38431667},
doi = {10.1038/s41467-024-46236-5},
url = {https://pub.dzne.de/record/268494},
}