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@ARTICLE{Jocher:277534,
author = {Jocher, Georg and Ozcelik, Gozde and Müller, Stephan A and
Hsia, Hung-En and Lastra Osua, Miranda and Hofmann, Laura I
and Aßfalg, Marlene and Dinkel, Lina and Feng, Xiao and
Schlepckow, Kai and Willem, Michael and Haass, Christian and
Tahirovic, Sabina and Blobel, Carl P and Lichtenthaler,
Stefan F},
title = {{T}he late-onset {A}lzheimer’s disease risk factor
{RHBDF}2 is a modifier of microglial {TREM}2 proteolysis},
journal = {Life science alliance},
volume = {8},
number = {5},
issn = {2575-1077},
address = {Heidelberg},
publisher = {EMBO Press},
reportid = {DZNE-2025-00430},
pages = {e202403080},
year = {2025},
abstract = {The cell surface receptor TREM2 is a key genetic risk
factor and drug target in Alzheimer’s disease (AD). In the
brain, TREM2 is expressed in microglia, where it undergoes
proteolytic cleavage, linked to AD risk, but the responsible
protease in microglia is still unknown. Another
microglial-expressed AD risk factor is catalytically
inactive rhomboid 2 (iRhom2, RHBDF2), which binds to and
acts as a non-catalytic subunit of the metalloprotease
ADAM17. A potential role in TREM2 proteolysis is not yet
known. Using microglial-like BV2 cells, bone
marrow–derived macrophages, and primary murine microglia,
we identify iRhom2 as a modifier of ADAM17-mediated TREM2
shedding. Loss of iRhom2 increased TREM2 in cell lysates and
at the cell surface and enhanced TREM2 signaling and
microglial phagocytosis of the amyloid β-peptide (Aβ).
This study establishes ADAM17 as a physiological TREM2
protease in microglia and suggests iRhom2 as a potential
drug target for modulating TREM2 proteolysis in AD.},
cin = {AG Lichtenthaler / AG Tahirovic / AG Haass},
ddc = {570},
cid = {I:(DE-2719)1110006 / I:(DE-2719)1140003 /
I:(DE-2719)1110007},
pnm = {352 - Disease Mechanisms (POF4-352)},
pid = {G:(DE-HGF)POF4-352},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:40081988},
doi = {10.26508/lsa.202403080},
url = {https://pub.dzne.de/record/277534},
}