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@INPROCEEDINGS{Bathe:283145,
author = {Bathe, Tim and Salomasova, Svetlana and Lalia, Manvir and
Kunze, Lea and Palumbo, Giovanna and Oos, Rosel and Joseph,
Emanuel and Brendel, Matthias},
title = {{M}ulti‐tracer {PET} monitoring of an immunomodulatory
therapy in 4{R} tauopathy: {E}valuating a novel drug's
impact on glial function and protein pathology},
journal = {Alzheimer's and dementia},
volume = {21},
number = {S2},
issn = {1552-5260},
reportid = {DZNE-2026-00041},
pages = {e104796},
year = {2025},
abstract = {The prevalence of neurodegenerative diseases (ND),
including Alzheimer's disease (AD) and non-AD tauopathies,
is projected to rise significantly by 2050 due to an aging
global population. Chronic neuroinflammation, driven by
glial activation in response to protein pathologies, is a
major contributor to disease progression. Targeting glial
dysfunction through immunomodulatory therapies offers a
promising approach to mitigate the effects of tauopathies
and other ND.PS19 mice receive chronic treatment with GV1001
over 5 months. Serial neuroimaging techniques, including PET
scans targeting tau protein, microglial activation, and
astrocytic responses, are employed to assess treatment
effects in vivo (Figure 1). Postmortem validation is
performed using immunohistochemistry and biochemical
methods, comparing treated mice to placebo and
non-transgenic controls.The research scope is to monitor the
efficacy of GV1001 in a transgenic tau mouse model (PS19)
with an early-intervention biomarker study using molecular
biology and neuroimaging techniques including TSPO
(microglia) PET, deprenyl (astroglia) PET, tau PET
(perfusion and retention) and CSF markers of inflammation
(e.g. sTREM2) and neurodegeneration (NfL). Preliminary
findings, expected to be presented at the conference, will
provide insights into the drug's ability to modulate glial
activity, restore homeostasis, and reduce tau pathology.This
study highlights the potential of monitoring
immunomodulatory strategies to address the complex interplay
between chronic neuroinflammation and protein aggregation in
ND. If successful, these findings could inform the
development of novel therapeutic approaches for AD and
related disorders, bridging the gap between preclinical
research and clinical application.},
month = {Jul},
date = {2025-07-27},
organization = {Alzheimer’s Association
International Conference, Toronto
(Canada), 27 Jul 2025 - 31 Jul 2025},
keywords = {Animals / Biomarkers: cerebrospinal fluid / Biomarkers:
metabolism / Mice / Mice, Transgenic / Disease Models,
Animal / Alzheimer Disease: drug therapy / Positron-Emission
Tomography / tau Proteins: metabolism / Humans / Brain:
metabolism / Brain: pathology / Brain: diagnostic imaging /
Brain: drug effects / Tauopathies: drug therapy / Microglia:
metabolism / Biomarkers (NLM Chemicals) / tau Proteins (NLM
Chemicals)},
cin = {AG Haass},
ddc = {610},
cid = {I:(DE-2719)1110007},
pnm = {352 - Disease Mechanisms (POF4-352)},
pid = {G:(DE-HGF)POF4-352},
typ = {PUB:(DE-HGF)1 / PUB:(DE-HGF)16},
doi = {10.1002/alz70856_104796},
url = {https://pub.dzne.de/record/283145},
}