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@ARTICLE{Zu:285042,
author = {Zu, Juan and Li, Cong and Cui, Mochen and Liu, Xinwu and
Pan, Zhouyang and Li, Xiaohe and Zhang, Fang and Gentz,
Johanna and Mitteregger-Kretzschmar, Gerda and Herms, Jochen
and Shi, Yuan},
title = {{P}ioglitazone attenuates complement-mediated microglial
synaptic engulfment in an {A}lzheimer's disease model.},
journal = {Brain},
volume = {149},
number = {2},
issn = {0006-8950},
address = {Oxford},
publisher = {Oxford Univ. Press},
reportid = {DZNE-2026-00166},
pages = {668 - 679},
year = {2026},
abstract = {Synaptic loss is an early hallmark of Alzheimer's disease
(AD), predominantly driven by aberrant microglial
reactivity. Pioglitazone, a peroxisome
proliferator-activated receptor gamma (PPAR-γ) agonist with
anti-diabetic properties, has been shown to suppress
microglial activity and improve cognitive performance in
both AD models and clinical studies. However, whether its
neuroprotective effects involve direct modulation of
synaptic architecture remains unclear. Here, using
longitudinal in vivo two-photon imaging, multi-channel
immunohistochemistry, super-resolution confocal microscopy
and three-dimensional reconstruction techniques in an AD
mouse model, we analyse synaptic and microglial
interactions. We show that a 4-week pioglitazone treatment
preserves dendritic spine density and enhances spine
stability over time. Mechanistically, pioglitazone reduces
synaptic C1q deposition, thereby limiting
complement-mediated microglial synaptic engulfment and
attenuating synapse loss. These findings identify
pioglitazone as a modulator of complement-dependent
microglial synaptic pruning and support its therapeutic
potential in preserving synaptic integrity during early AD
pathogenesis.},
keywords = {Pioglitazone: pharmacology / Animals / Alzheimer Disease:
drug therapy / Alzheimer Disease: pathology / Alzheimer
Disease: metabolism / Microglia: drug effects / Microglia:
metabolism / Microglia: pathology / Mice / Synapses: drug
effects / Synapses: pathology / Disease Models, Animal /
Mice, Transgenic / Dendritic Spines: drug effects /
Dendritic Spines: pathology / Complement C1q: metabolism /
Mice, Inbred C57BL / Male / PPAR gamma: agonists / Humans /
Alzheimer’s disease (Other) / microglia (Other) /
peroxisome proliferator-activated receptor-γ (Other) /
pioglitazone (Other) / synaptic plasticity (Other) /
Pioglitazone (NLM Chemicals) / Complement C1q (NLM
Chemicals) / PPAR gamma (NLM Chemicals)},
cin = {AG Herms},
ddc = {610},
cid = {I:(DE-2719)1110001},
pnm = {352 - Disease Mechanisms (POF4-352)},
pid = {G:(DE-HGF)POF4-352},
typ = {PUB:(DE-HGF)16},
pubmed = {pmid:41396874},
doi = {10.1093/brain/awaf462},
url = {https://pub.dzne.de/record/285042},
}